Elucirem™ (gadopiclenol) has a high kinetic stability with a comparable safety profile to gadobutrol2-4

 


Elucirem™ has at least 4 x the kinetic stability of approved GBCAs1

The macrocyclic structure of Elucirem™ is associated with higher kinetic stability and a longer dissociation half-life1

Elucirem™ (gadopiclenol) has been shown to have a comparable safety profile to gadobutrol in clinical trials2-4

•  In the PICTURE trial, treatment emergent adverse event (TEAE) incidence was 14.6% after MRI with gadopiclenol and 17.6% after MRI with gadobutrol.3,4
•  In the PROMISE trial, TEAE incidence was 18.1% after MRI with gadopiclenol and 20.0% after MRI with gadobutrol.3,4

At least one TEAE related to contrast agent in phase III clinical trial3,4

 

Elucirem™ (gadopiclenol)
Rate (%)

Gadovist® (gadobutrol)
Rate (%)

CNS MRI (PICTURE trial) 4.9% 15 reported in 12 patients 6.9% 19 reported in 17 patients
Body MRI (PROMISE trial) 4.2% 14 reported in 12 patients 5.5% 19 reported in 16 patients

 

Adverse reactions reported in 0.2% of patients (2 years to 88 years old) who received the recommended dose of Elucirem™ (0.05 mmol/kg) in clinical trials3,4

Reaction

Rate (%)

Injection site pain  0,7
Headache 0,7
Nausea 0,4
Injection site warmth 0,4
Injection site coldness 0,3
Dizziness 0,3
Localised swelling 0,3


The table lists adverse reactions that occurred in >0.2% of patients who received 0.05 mmol/kg Elucirem™
 

No cases of nephrogenic systemic fibrosis have been reported in clinical trials with Elucirem™1
 

Discover the simple dosing and administration of Elucirem™

Trademarks are the property of their respective owners.

CNS: Central Nervous System
GBCA: Gadolinium-Based Contrast Agent
MRI: Magnetic Resonance Imaging NSF: Nephrogenic Systemic Fibrosis
TEAE: Treatment Emergent Adverse Events

 

References

1. Robic C, Port M, Rousseaux O, et al. Physicochemical and Pharmacokinetic Profiles of Gadopiclenol: A New Macrocyclic Gadolinium Chelate With High T1 Relaxivity. Invest Radiol. 2019 Aug;54(8):475-484.
2. Elucirem Summary of Product Characteristics. 2023.
3. Loevner LA, Kolumban B, Hutóczki G, et al. Efficacy and Safety of Gadopiclenol for Contrast-Enhanced MRI of the Central Nervous System: The PICTURE Randomized Clinical Trial. Invest Radiol. 2023 May 1;58(5):307-313.
4. Kuhl C, Csőszi T, Piskorski W, et al. Efficacy and safety of half-dose gadopiclenol versus full-dose gadobutrol for contrast-enhanced body MRI. Radiology. 2023 Jul;308(1):e222612.

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